UPSC MainsBOTANY-PAPER-II202410 Marks
Q3.

Discuss what are cell receptors and how do they help in cell signalling? Elaborate the answer with the help of at least one example.

How to Approach

This question requires a detailed understanding of cell receptors and their role in cell signaling. The answer should begin with defining cell receptors and outlining the general principles of cell signaling. It should then elaborate on different types of receptors and their mechanisms of action. Finally, a specific example, like insulin signaling, should be used to illustrate the process. A clear, structured approach with appropriate biological terminology is crucial for a good score.

Model Answer

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Introduction

Cell signaling is fundamental to life, enabling cells to perceive and respond to their environment. This intricate communication relies heavily on **cell receptors**, specialized proteins located on the cell surface or within the cell. These receptors act as gatekeepers, binding to signaling molecules (ligands) and initiating a cascade of events that ultimately alter cellular function. Understanding cell receptors and their signaling pathways is crucial for comprehending various biological processes, from development and immunity to disease pathogenesis. This answer will discuss the nature of cell receptors, their role in cell signaling, and illustrate the process with the example of insulin signaling.

What are Cell Receptors?

Cell receptors are proteins that bind to specific signaling molecules, also known as ligands. This binding event initiates a conformational change in the receptor, triggering a series of intracellular events. Receptors can be broadly classified based on their location and mechanism of action:

  • Cell-Surface Receptors: These receptors span the cell membrane and bind to hydrophilic ligands that cannot easily cross the plasma membrane. Examples include G protein-coupled receptors (GPCRs), receptor tyrosine kinases (RTKs), and ligand-gated ion channels.
  • Intracellular Receptors: These receptors are located within the cytoplasm or nucleus and bind to hydrophobic ligands that can diffuse across the cell membrane, such as steroid hormones.

How do Cell Receptors Help in Cell Signaling?

Cell signaling involves a series of steps:

  1. Reception: The ligand binds to the receptor.
  2. Transduction: The binding event activates intracellular signaling pathways, often involving a cascade of protein kinases.
  3. Response: The signaling pathway ultimately leads to a cellular response, such as changes in gene expression, enzyme activity, or cell shape.

Types of Cell Signaling Pathways

  • GPCR Signaling: Ligand binding activates a G protein, which then activates or inhibits an effector protein, leading to a cellular response.
  • RTK Signaling: Ligand binding causes receptor dimerization and autophosphorylation, creating docking sites for intracellular signaling proteins.
  • Intracellular Receptor Signaling: Ligand binding causes the receptor to translocate to the nucleus and regulate gene expression.

Example: Insulin Signaling

Insulin signaling is a classic example of receptor-mediated cell signaling. Insulin, a peptide hormone, binds to the insulin receptor (an RTK) on the surface of target cells, such as muscle and fat cells.

The steps involved are:

  1. Insulin binds to the insulin receptor, causing it to dimerize and autophosphorylate.
  2. The phosphorylated receptor recruits intracellular signaling proteins, such as IRS (insulin receptor substrate).
  3. IRS activates downstream signaling pathways, including the PI3K/Akt pathway and the MAPK pathway.
  4. These pathways lead to increased glucose uptake, glycogen synthesis, and protein synthesis.

Dysregulation of insulin signaling can lead to insulin resistance and type 2 diabetes.

Component Role in Insulin Signaling
Insulin Receptor Binds insulin and initiates the signaling cascade.
IRS Recruited by the activated receptor and activates downstream pathways.
PI3K/Akt Pathway Promotes glucose uptake and glycogen synthesis.
MAPK Pathway Stimulates cell growth and proliferation.

Conclusion

Cell receptors are essential components of cell signaling, enabling cells to respond to their environment and maintain homeostasis. Understanding the different types of receptors and their signaling pathways is crucial for comprehending a wide range of biological processes and diseases. The example of insulin signaling illustrates the complexity and importance of receptor-mediated cell communication. Further research into cell receptors and their signaling mechanisms will undoubtedly lead to new therapeutic strategies for various diseases.

Answer Length

This is a comprehensive model answer for learning purposes and may exceed the word limit. In the exam, always adhere to the prescribed word count.

Additional Resources

Key Definitions

Ligand
A molecule that binds to a receptor, initiating a biological response.
Autophosphorylation
The process by which a kinase adds a phosphate group to itself, often activating the kinase and creating docking sites for other proteins.

Key Statistics

Approximately 34% of all approved drugs target G protein-coupled receptors (GPCRs), making them the largest class of drug targets.

Source: Pharmacological Reviews, 2018

It is estimated that over 400 different receptor types exist in the human genome.

Source: Nature Reviews Drug Discovery, 2010 (Knowledge Cutoff)

Examples

Nicotinic Acetylcholine Receptor

This ligand-gated ion channel is crucial for neuromuscular transmission. Binding of acetylcholine opens the channel, allowing ions to flow and triggering muscle contraction.

Frequently Asked Questions

What happens if a receptor is mutated?

Mutations in receptors can alter their binding affinity for ligands, their signaling efficiency, or their localization within the cell. This can lead to a variety of diseases, depending on the specific receptor and mutation.