UPSC MainsMEDICAL-SCIENCE-PAPER-II20183 Marks
Q8.

Enumerate the side effects of commonly used anti-psychotic drugs.

How to Approach

This question requires a detailed understanding of pharmacovigilance concerning antipsychotic drugs. The answer should systematically enumerate the side effects, categorizing them for clarity (e.g., neurological, metabolic, cardiovascular). Mentioning specific antipsychotic classes and their associated side effect profiles will demonstrate depth. A structured approach, perhaps using subheadings for each category of side effects, is recommended. Focus on commonly used drugs and their well-documented adverse effects.

Model Answer

0 min read

Introduction

Antipsychotic drugs are a cornerstone in the treatment of psychotic disorders like schizophrenia and bipolar disorder. These medications work by modulating dopamine and serotonin neurotransmission in the brain, alleviating symptoms such as hallucinations and delusions. However, their use is often accompanied by a range of side effects, stemming from their broad pharmacological actions. Understanding these adverse effects is crucial for clinicians to optimize treatment, minimize patient distress, and ensure adherence to therapy. This answer will enumerate the side effects of commonly used antipsychotic drugs, categorized for clarity and comprehensiveness.

Neurological Side Effects

Neurological side effects are among the most common and clinically significant adverse effects associated with antipsychotic medications.

  • Extrapyramidal Symptoms (EPS): These include dystonia (sustained muscle contractions), akathisia (restlessness), parkinsonism (tremor, rigidity, bradykinesia), and tardive dyskinesia (involuntary movements, often of the face and tongue). First-generation antipsychotics (FGAs) like haloperidol are more strongly associated with EPS due to their potent dopamine D2 receptor blockade.
  • Neuroleptic Malignant Syndrome (NMS): A rare but life-threatening complication characterized by fever, muscle rigidity, altered mental status, and autonomic instability. Requires immediate medical intervention.
  • Seizures: Antipsychotics can lower the seizure threshold, increasing the risk of seizures, particularly in individuals with pre-existing seizure disorders.

Metabolic Side Effects

Second-generation antipsychotics (SGAs) like olanzapine, clozapine, and quetiapine are more frequently associated with metabolic disturbances.

  • Weight Gain: Significant weight gain is common, contributing to obesity and related health problems.
  • Dyslipidemia: Increases in cholesterol and triglyceride levels.
  • Hyperglycemia and Diabetes Mellitus: Antipsychotics can impair glucose metabolism, increasing the risk of developing type 2 diabetes.
  • Metabolic Syndrome: A cluster of conditions including abdominal obesity, high blood pressure, high blood sugar, and abnormal cholesterol levels.

Cardiovascular Side Effects

Antipsychotics can have various effects on the cardiovascular system.

  • QT Prolongation: Some antipsychotics (e.g., thioridazine, ziprasidone) can prolong the QT interval on an electrocardiogram, increasing the risk of torsades de pointes, a potentially fatal arrhythmia.
  • Orthostatic Hypotension: A sudden drop in blood pressure upon standing, leading to dizziness and falls.
  • Increased Risk of Stroke: Particularly in elderly patients with dementia-related psychosis.

Anticholinergic Side Effects

These effects are more prominent with certain antipsychotics.

  • Dry Mouth: Reduced saliva production.
  • Constipation: Decreased gastrointestinal motility.
  • Blurred Vision: Impaired accommodation.
  • Urinary Retention: Difficulty emptying the bladder.

Other Side Effects

  • Sedation: Many antipsychotics cause drowsiness and fatigue.
  • Sexual Dysfunction: Decreased libido, erectile dysfunction, and menstrual irregularities.
  • Prolactin Elevation: Some antipsychotics (e.g., risperidone, paliperidone) can increase prolactin levels, leading to gynecomastia (breast enlargement in males), galactorrhea (milk production), and menstrual irregularities in females.
  • Agranulocytosis: A rare but serious side effect associated with clozapine, characterized by a severe reduction in white blood cells, increasing the risk of infection. Requires regular blood monitoring.
Antipsychotic Class Common Side Effects
First-Generation (FGAs) EPS, Tardive Dyskinesia, Hyperprolactinemia
Second-Generation (SGAs) Metabolic Syndrome, Weight Gain, Dyslipidemia, Hyperglycemia
Clozapine Agranulocytosis, Sedation, Weight Gain, Seizures

Conclusion

Antipsychotic drugs, while effective in managing psychotic disorders, are associated with a wide spectrum of side effects. These range from relatively mild inconveniences like sedation and dry mouth to potentially life-threatening complications like NMS and agranulocytosis. Careful monitoring, individualized treatment plans, and patient education are essential to minimize risks and optimize therapeutic outcomes. Ongoing research continues to refine our understanding of these side effects and develop strategies for their prevention and management.

Answer Length

This is a comprehensive model answer for learning purposes and may exceed the word limit. In the exam, always adhere to the prescribed word count.

Additional Resources

Key Definitions

Pharmacovigilance
The science and activities relating to the detection, assessment, understanding and prevention of adverse effects or any other drug-related problem.
Tardive Dyskinesia
A movement disorder characterized by involuntary, repetitive movements, often affecting the face, tongue, and limbs, that can develop after prolonged use of dopamine-blocking agents like antipsychotics.

Key Statistics

Approximately 20-30% of patients with schizophrenia discontinue antipsychotic medication within the first year due to side effects.

Source: American Psychiatric Association (2013)

The prevalence of tardive dyskinesia in patients treated with first-generation antipsychotics is estimated to be around 20-30% after long-term use.

Source: National Institute of Mental Health (NIMH) - Knowledge cutoff 2023

Examples

Olanzapine and Weight Gain

Olanzapine is known for its high propensity to cause significant weight gain, often leading to metabolic syndrome and increased cardiovascular risk in patients.

Frequently Asked Questions

Can side effects be managed?

Yes, many side effects can be managed through dose adjustments, switching medications, or adding other medications to counteract the adverse effects (e.g., anticholinergics for EPS, metformin for metabolic syndrome).