UPSC MainsMEDICAL-SCIENCE-PAPER-I20255 Marks
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Q48.

Name the drugs, doses and duration of treatment after post-exposure prophylaxis of HIV.

How to Approach

To answer this question effectively, one should define HIV Post-Exposure Prophylaxis (PEP) and emphasize the importance of timely administration. The core of the answer will detail the recommended drug regimens, including specific drug names, their standard doses, and the duration of treatment, referencing the latest guidelines from authoritative bodies like WHO and national organizations. It is crucial to highlight variations based on the type of exposure (occupational vs. non-occupational) and special considerations.

Model Answer

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Introduction

Post-Exposure Prophylaxis (PEP) for HIV is an emergency medical intervention involving the administration of antiretroviral (ARV) drugs to prevent HIV infection after potential exposure to the virus. It is a critical component of HIV prevention strategies, particularly in occupational settings (e.g., needlestick injuries for healthcare workers) and non-occupational settings (e.g., unprotected sexual contact, sexual assault). The efficacy of PEP is highly time-dependent, with guidelines emphasizing initiation as soon as possible, ideally within 24 hours and no later than 72 hours post-exposure. The goal is to interrupt the early stages of viral replication before the virus can establish a permanent infection.

Drugs, Doses, and Duration of Treatment for HIV Post-Exposure Prophylaxis (PEP)

The choice of antiretroviral (ARV) drugs, their dosages, and the duration of treatment for HIV Post-Exposure Prophylaxis (PEP) are guided by international and national health organizations, primarily the World Health Organization (WHO) and national bodies like India's National AIDS Control Organisation (NACO). These guidelines are regularly updated to reflect advancements in ARV therapies, aiming for increased efficacy, reduced side effects, and improved accessibility.

Key Principles of PEP Administration:

  • Timeliness: PEP must be initiated as soon as possible after exposure, ideally within 24 hours, and definitely within 72 hours. Delay significantly reduces its effectiveness.
  • Duration: The standard duration of PEP treatment is 28 days (4 weeks).
  • Regimen: A three-drug regimen is generally preferred over a two-drug regimen for optimal effectiveness.
  • Assessment: A thorough risk assessment is crucial, considering the type of exposure and the HIV status of the source.

Recommended PEP Regimens (General Guidelines - WHO and recent updates):

Recent guidelines, including updates from the US CDC (May 2025) and WHO (July 2024), favor newer, well-tolerated antiretroviral drugs. While specific national guidelines might have slight variations, the core components remain consistent.

Preferred Regimens for Adults and Adolescents:

The current preferred regimens typically include a combination of two Nucleoside/Nucleotide Reverse Transcriptase Inhibitors (NRTIs) and one Integrase Strand Transfer Inhibitor (INSTI).

  • Option 1 (WHO, US CDC 2025 preferred):
    • Drugs: Bictegravir (BIC) + Emtricitabine (FTC) + Tenofovir Alafenamide (TAF)
      (often available as a single fixed-dose combination pill)
    • Dose: BIC 50 mg / FTC 200 mg / TAF 25 mg, once daily
    • Duration: 28 days
  • Option 2 (WHO, US CDC 2025 preferred; also widely recommended):
    • Drugs: Dolutegravir (DTG) + Emtricitabine (FTC) or Lamivudine (3TC) + Tenofovir Disoproxil Fumarate (TDF) or Tenofovir Alafenamide (TAF)
    • Dose: DTG 50 mg once daily, plus FTC 200 mg once daily or 3TC 300 mg once daily, plus TDF 300 mg once daily or TAF 25 mg once daily. (Often combined into 2 pills: DTG + FDC of TDF/FTC or TAF/FTC)
    • Duration: 28 days

Older/Alternative Regimens (Still used in some contexts, or where preferred regimens are not available):

Previous guidelines often recommended regimens including Efavirenz (EFV) or ritonavir-boosted protease inhibitors (PI/r).

  • NACO (India) 2014 Guidelines (Still widely referred to in India, though newer WHO/CDC guidelines may be incorporated):
    • Drugs: Tenofovir (TDF) + Lamivudine (3TC) + Efavirenz (EFV)
    • Dose: TDF 300 mg + 3TC 300 mg + EFV 600 mg, once daily (often as a single fixed-dose combination pill, TLD)
    • Duration: 28 days
    • Note: If intolerance to Efavirenz, a regimen containing Tenofovir + Lamivudine + Protease Inhibitor (e.g., Atazanavir/ritonavir (ATV/r) or Lopinavir/ritonavir (LPV/r)) can be used after expert consultation.

Considerations for Special Populations:

  • Children: Regimens and dosages are adjusted based on age and weight bands, often involving combinations like Abacavir (ABC) + Lamivudine (3TC) + Lopinavir/ritonavir (LPV/r) or Zidovudine (ZDV) + 3TC + LPV/r, or ABC + 3TC + DTG.
  • Pregnancy and Breastfeeding: Specific ARV drugs are preferred based on safety profiles during pregnancy and breastfeeding. Dolutegravir-based regimens are generally recommended, with careful consideration and expert consultation.
  • Source on ART or with potential drug resistance: Expert consultation is crucial to select a regimen less likely to be affected by potential drug resistance in the source.

Table: Summary of Key PEP Regimens and Duration

Regimen Type Drugs (Examples) Typical Doses Duration Key Considerations
Preferred (WHO/US CDC 2025) Bictegravir/Emtricitabine/Tenofovir Alafenamide (BIC/FTC/TAF) One fixed-dose combination pill daily 28 days High efficacy, good tolerability. Often a single pill simplifies adherence.
Preferred (WHO/US CDC 2025) Dolutegravir (DTG) + FDC of Tenofovir (TDF/TAF) / Emtricitabine (FTC) or Lamivudine (3TC) DTG 50mg OD + FDC (e.g., TDF 300mg/FTC 200mg) OD 28 days Highly effective, widely available.
Older/Alternative (e.g., NACO 2014) Tenofovir (TDF) + Lamivudine (3TC) + Efavirenz (EFV) TDF 300mg OD + 3TC 300mg OD + EFV 600mg OD (often FDC) 28 days Effective, but EFV can have CNS side effects. Not recommended for two-drug regimens.

Monitoring and Follow-up: After initiating PEP, individuals undergo baseline HIV testing and other relevant blood tests. Follow-up HIV testing (e.g., at 4-6 weeks and 12 weeks post-exposure) is critical to determine the success of PEP. Counseling on adherence to the regimen, potential side effects, and ongoing risk reduction strategies (including transition to Pre-Exposure Prophylaxis, PrEP, if at ongoing risk) are integral parts of the PEP management protocol.

Conclusion

HIV Post-Exposure Prophylaxis (PEP) is a vital intervention for preventing HIV infection after potential exposure, contingent on rapid initiation and strict adherence to the regimen. The current standard involves a 28-day course of a three-drug antiretroviral combination, with preferred options generally including an integrase inhibitor (like bictegravir or dolutegravir) alongside two NRTIs. Adherence to these guidelines, coupled with comprehensive counseling and follow-up, significantly reduces the risk of HIV transmission. Continuous updates in guidelines aim to improve drug efficacy, reduce side effects, and enhance accessibility, reflecting the evolving landscape of HIV prevention and treatment.

Answer Length

This is a comprehensive model answer for learning purposes and may exceed the word limit. In the exam, always adhere to the prescribed word count.

Additional Resources

Key Definitions

Post-Exposure Prophylaxis (PEP)
PEP is the short-term use of antiretroviral drugs to reduce the likelihood of HIV infection after potential exposure to the virus, such as through unprotected sex, needlestick injuries, or sexual assault.
Fixed-Dose Combination (FDC)
An FDC is a combination of two or more active pharmaceutical ingredients combined in a single dosage form. This simplifies drug regimens, improves adherence, and reduces pill burden for patients.

Key Statistics

PEP is most effective when initiated within 24 hours of exposure. Its effectiveness significantly decreases if started beyond 72 hours, with some studies suggesting little to no benefit after this critical window.

Source: WHO Guidelines for HIV Post-Exposure Prophylaxis (July 2024), US CDC Guidelines for PEP (May 2025)

Despite advancements in testing and treatment, over one million people became infected with HIV globally in 2022, underscoring the continued importance of prevention strategies like PEP.

Source: WHO Guidelines for HIV Post-Exposure Prophylaxis (July 2024)

Examples

Occupational Exposure PEP

A healthcare worker accidentally pricks their finger with a needle used on an HIV-positive patient. Immediate reporting and initiation of a 28-day course of a three-drug PEP regimen (e.g., Dolutegravir + TDF/FTC) within hours of the incident is crucial to prevent potential HIV transmission.

Non-Occupational Exposure PEP

An individual has unprotected sexual intercourse with a partner of unknown HIV status or a known HIV-positive partner with a detectable viral load. Seeking medical attention within 72 hours to assess risk and potentially begin PEP is a critical step in preventing HIV infection.

Frequently Asked Questions

Can PEP be used more than 72 hours after exposure?

While PEP is ideally started within 24 hours and definitely within 72 hours, its effectiveness significantly diminishes after 72 hours. Current guidelines generally do not recommend initiating PEP beyond this window as the likelihood of preventing infection becomes very low. However, individual risk assessment by a clinician is always paramount.

Is a two-drug PEP regimen effective?

While a two-drug regimen can have some effectiveness, current international and national guidelines (like WHO and NACO 2014) strongly prefer and recommend a three-drug regimen for HIV PEP due to its superior efficacy in preventing HIV infection. Two-drug regimens are generally no longer recommended for PEP in most situations.

Topics Covered

Infectious DiseasesPharmacologyPublic HealthHIV/AIDSAntiretroviral DrugsPreventive Medicine